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Treatment Most patients with clenbuterol toxicity can be managed with supportive therapy, including IV fluids, potassium supplementation, and benzodiazepines for agitation. For patients who are very tachycardic or hypotensive, β-blockers such as metoprolol, labetalol, or esmolol, can be used to counteract the β-agonism of the clenbuterol. Dosage Takeaway Clenbuterol is a substance best known for its use in treating asthma and encouraging weight loss. It is not available for humans in the United States. Treatment of overdose is simple and should be promptly started using in-travenous fluid hydration and potassium supplementation. Benzodiazepines may be utilized for agitation or delirium. Β-blockers or phenylephrine may be used to give hemodynamic support. PMID: 18072161 PMCID: PMC3550084 DOI: 10. 1007/BF03160909 Abstract Objective: We are presenting a case illustrating the complex metabolic and rhythm disturbances associated with acute clenbuterol intoxication. Background: Clenbuterol is a long-acting beta2-adrenergic agonist primarily used in veterinary medicine in the United States. Dosage Risks and side effects Current research Outlook Clenbuterol has approval for human use as an asthma drug in some countries but is banned for this use in the United States. Management of clenbuterol overdose is supportive care. There is no antidote. Sedatives or anxiolytics may be used to treat agitation or psychosis, and β-blockers may be administered in hemodynamic compromise or myocardial infarction as long as concomitant cocaine ingestion has been ruled out
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